This volume presents cutting-edge chemical and molecular strategies. Chapters detail bioorthogonal cycloadditions, electrophiles, self-labeling systems, noncanonical amino acids, site-selective bioconjugation across proteins, nucleic acids, cells, and viral assemblies. Written in the highly successful Methods in Molecular Biology series format, chapters include introductions to their respective topics, lists of the necessary materials and reagents, step-by-step, readily reproducible laboratory protocols, and tips on troubleshooting and avoiding known pitfalls. Cutting-edge and thorough, Bioconjugation Methods is a valuable resource for all researchers who are looking to learn more about this important and advancing field.